| 1 |
CC-1065 and the Duocarmycins - Synthetic Studies
Boger DL, Boyce CW, Garbaccio RM, Goldberg JA
Chemical Reviews, 97(3), 787, 1997 |
| 2 |
Total Synthesis of (+)-Duocarmycin-A, EPI-(+)-Duocarmycin-A and Their Unnatural Enantiomers - Assessment of Chemical and Biological Properties
Boger DL, Mckie JA, Nishi T, Ogiku T
Journal of the American Chemical Society, 119(2), 311, 1997 |
| 3 |
Duocarmycin SA Shortened, Simplified, and Extended Agents - A Systematic Examination of the Role of the DNA-Binding Subunit
Boger DL, Hertzog DL, Bollinger B, Johnson DS, Cai H, Goldberg J, Turnbull P
Journal of the American Chemical Society, 119(21), 4977, 1997 |
| 4 |
Synthesis, X-Ray Structure, and Properties of Fluorocyclopropane Analogs of the Duocarmycins Incorporating the 9,9-Difluoro-1,2,9,9A-Tetrahydrocyclopropa(C)Benzo(E)Indol-4-One (F2Cbi) Alkylation Subunit
Boger DL, Jenkins TJ
Journal of the American Chemical Society, 118(37), 8860, 1996 |
| 5 |
2nd Definitive Test of Proposed Models for the Origin of the CC-1065 and Duocarmycin DNA Alkylation Selectivity
Boger DL, Johnson DS
Journal of the American Chemical Society, 117(4), 1443, 1995 |
| 6 |
DNA Alkylation Properties of CC-1065 and Duocarmycin Analogs Incorporating the 2,3,10,10A-Tetrahydrocyclopropa(D)Benzo(F)Quinol-5-One Alkylation Subunit - Identification of Subtle Structural Features That Contribute to the Regioselectivity of the Adenine N3 Alkylation Reaction
Boger DL, Mesini P
Journal of the American Chemical Society, 117(47), 11647, 1995 |
| 7 |
(+)- and ENT-(-)-Duocarmycin SA and (+)- and ENT-(-)-N-BOC-DSA DNA Alkylation Properties - Alkylation Site Models That Accommodate the Offset at-Rich Adenine N3 Alkylation Selectivity of the Enantiomeric Agents
Boger DL, Johnson DS, Yun WY
Journal of the American Chemical Society, 116(5), 1635, 1994 |
| 8 |
Role of the CC-1065 and Duocarmycin N-2 Substituent - Validation of a Direct Relationship Between Solvolysis Chemical-Stability and in-Vitro Biological Potency
Boger DL, Yun WY
Journal of the American Chemical Society, 116(12), 5523, 1994 |
| 9 |
Chemical and Structural Comparison of N-BOC-Cbq and N-BOC-CBI - Identification and Structural Origin of an Unappreciated But Productive Stability of the CC-1065 and Duocarmycin SA Alkylation Subunits
Boger DL, Mesini P, Tarby CM
Journal of the American Chemical Society, 116(14), 6461, 1994 |
| 10 |
Acid-Dependent Electrophilicity of Cyclopropylpyrroloindoles - Natures Masking Strategy for a Potent DNA Alkylator
Warpehoski MA, Harper DE
Journal of the American Chemical Society, 116(17), 7573, 1994 |
