검색결과 : 10건
| No. | Article |
|---|---|
| 1 |
Apralogs: Apramycin 5-O-Glycosides and Ethers with Improved Antibacterial Activity and Ribosomal Selectivity and Reduced Susceptibility to the Aminoacyltranserferase (3)-IV Resistance Determinant Quirke JCK, Rajasekaran P, Sarpe V, Sonousi A, Osinnii I, Gysin M, Haldimann K, Fang QJ, Shcherbakov D, Hobbie SN, Sha SH, Schacht J, Vasella A, Bottger EC, Crich D Journal of the American Chemical Society, 142(1), 530, 2020 |
| 2 |
Design, Multigram Synthesis, and in Vitro and in Vivo Evaluation of Propylamycin: A Semisynthetic 4,5-Deoxystreptamine Class Aminoglycoside for the Treatment of Drug-Resistant Enterobacteriaceae and Other Gram-Negative Pathogens Matsushita T, Sati GC, Kondasinghe N, Pirrone MG, Kato T, Waduge P, Kumar HS, Sanchon AC, Dobosz-Bartoszek M, Shcherbakov D, Juhas M, Hobbie SN, Schrepfer T, Chow CS, Polikanov YS, Schacht J, Vasella A, Bottger EC, Crich D Journal of the American Chemical Society, 141(12), 5051, 2019 |
| 3 |
Structure-Based Design and Synthesis of Apramycin-Paromomycin Analogues: Importance of the Configuration at the 6 '-Position and Differences between the 6 '-Amino and Hydroxy Series Mandhapati AR, Yang GY, Kato T, Shcherbakov D, Hobbie SN, Vasella A, Bottger EC, Crich D Journal of the American Chemical Society, 139(41), 14611, 2017 |
| 4 |
Influence of 4'-O-Glycoside Constitution and Configuration on Ribosomal Selectivity of Paromomycin Matsushita T, Chen WW, Juskeviciene R, Teo YJ, Shcherbakov D, Vasella A, Bottger EC, Crich D Journal of the American Chemical Society, 137(24), 7706, 2015 |
| 5 |
Glycosidase inhibition: An assessment of the binding of 18 putative transition-state mimics Gloster TM, Meloncelli P, Stick RV, Zechel D, Vasella A, Davies GJ Journal of the American Chemical Society, 129(8), 2345, 2007 |
| 6 |
Probing specific lectin-carbohydrate interactions using atomic force microscopy imaging and force measurements Touhami A, Hoffmann B, Vasella A, Denis FA, Dufrene YF Langmuir, 19(5), 1745, 2003 |
| 7 |
The active site of cellobiohydrolase Cel6A from Trichoderma reesei: The roles of aspartic acids D221 and D175 Koivula A, Ruohonen L, Wohlfahrt G, Reinikainen T, Teeri TT, Piens K, Claeyssens M, Weber M, Vasella A, Becker D, Sinnott ML, Zou JY, Kleywegt GJ, Szardenings M, Stahlberg J, Jones TA Journal of the American Chemical Society, 124(34), 10015, 2002 |
| 8 |
Lateral protonation of a glycosidase inhibitor. Structure of the Bacillus agaradhaerens Cel5A in complex with a cellobiose-derived imidazole at 0.97 angstrom resolution Varrot A, Schulein M, Pipelier M, Vasella A, Davies GJ Journal of the American Chemical Society, 121(11), 2621, 1999 |
| 9 |
Synthesis and enzymatic phosphorylation of a photoactivatable dolichol analogue Grassi D, Lippuner V, Aebi M, Brunner J, Vasella A Journal of the American Chemical Society, 119(45), 10992, 1997 |
| 10 |
Self-Assembled Hexasaccharides - Surface Characterization of Thiol-Terminated Sugars Adsorbed on a Gold Surface Fritz MC, Hahner G, Spencer ND, Burli R, Vasella A Langmuir, 12(25), 6074, 1996 |